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Title | Design, synthesis and biological evaluations of N-Hydroxy thienopyrimidine-2,4-diones as inhibitors of HIV reverse transcriptase-associated RNase H. |
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Journal, issue, pages | Eur J Med Chem, Vol. 141, Page 149-161, Year 2017 |
Publish date | Aug 15, 2017 (structure data deposition date) |
Authors | Kankanala, J. / Kirby, K.A. / Huber, A.D. / Casey, M.C. / Wilson, D.J. / Sarafianos, S.G. / Wang, Z. |
External links | Eur J Med Chem / PubMed:29031062 |
Methods | X-ray diffraction |
Resolution | 1.8 Å |
Structure data | PDB-6aoc: |
Chemicals | ChemComp-MN: ChemComp-ZW2: ChemComp-PGE: ChemComp-EDO: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / TRANSFERASE INHIBITOR / HIV-1 / TRANSFERASE - TRANSFERASE INHIBITOR complex |