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-Structure paper
Title | Absolute Binding Free Energy Calculation and Design of a Subnanomolar Inhibitor of Phosphodiesterase-10. |
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Journal, issue, pages | J. Med. Chem., Vol. 62, Page 2099-2111, Year 2019 |
Publish date | Apr 9, 2018 (structure data deposition date) |
![]() | Li, Z. / Huang, Y. / Wu, Y. / Chen, J. / Wu, D. / Zhan, C.G. / Luo, H.B. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.8 Å |
Structure data | ![]() PDB-5znl: |
Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-MG: ![]() ChemComp-9G6: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE / PDE10A inhibitor |