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-Structure paper
Title | TAK-137, an AMPA-R potentiator with little agonistic effect, has a wide therapeutic window. |
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Journal, issue, pages | Neuropsychopharmacology, Vol. 44, Page 961-970, Year 2019 |
Publish date | Mar 7, 2018 (structure data deposition date) |
![]() | Kunugi, A. / Tanaka, M. / Suzuki, A. / Tajima, Y. / Suzuki, N. / Suzuki, M. / Nakamura, S. / Kuno, H. / Yokota, A. / Sogabe, S. ...Kunugi, A. / Tanaka, M. / Suzuki, A. / Tajima, Y. / Suzuki, N. / Suzuki, M. / Nakamura, S. / Kuno, H. / Yokota, A. / Sogabe, S. / Kosugi, Y. / Awasaki, Y. / Kaku, T. / Kimura, H. |
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Methods | X-ray diffraction |
Resolution | 1.25 - 1.65 Å |
Structure data | ![]() PDB-5zg0: ![]() PDB-5zg1: ![]() PDB-5zg2: ![]() PDB-5zg3: |
Chemicals | ![]() ChemComp-GLU: ![]() ChemComp-ZN: ![]() ChemComp-9C3: ![]() ChemComp-ACT: ![]() ChemComp-HOH: ![]() ChemComp-9C0: ![]() ChemComp-SO4: ![]() ChemComp-GOL: ![]() ChemComp-ZK1: ![]() ChemComp-9C6: |
Source |
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![]() | TRANSPORT PROTEIN / AMPA RECEPTOR LIGAND-BINDING DOMAIN / ALLOSTERIC MODULATION COMPLEX / MEMBRANE PROTEIN |