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-Structure paper
Title | Development and evaluation of a novel series of Nitroxoline-derived BET inhibitors with antitumor activity in renal cell carcinoma. |
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Journal, issue, pages | Oncogenesis, Vol. 7, Page 83-83, Year 2018 |
Publish date | Jan 20, 2018 (structure data deposition date) |
Authors | Chen, W. / Zhang, H. / Chen, Z. / Jiang, H. / Liao, L. / Fan, S. / Xing, J. / Xie, Y. / Chen, S. / Ding, H. ...Chen, W. / Zhang, H. / Chen, Z. / Jiang, H. / Liao, L. / Fan, S. / Xing, J. / Xie, Y. / Chen, S. / Ding, H. / Chen, K. / Luo, C. / Zheng, M. / Yao, Z. / Huang, Y. / Zhang, Y. |
External links | Oncogenesis / PubMed:30385738 |
Methods | X-ray diffraction |
Resolution | 1.631 - 1.991 Å |
Structure data | PDB-5z5t: PDB-5z5u: PDB-5z5v: |
Chemicals | ChemComp-96R: ChemComp-HOH: ChemComp-96U: ChemComp-96X: |
Source |
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Keywords | TRANSCRIPTION/INHIBITOR / BRD4 / Inhibitor / Complex / PROTEIN BINDING / TRANSCRIPTION-INHIBITOR complex |