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-Structure paper
Title | Y08060: A Selective BET Inhibitor for Treatment of Prostate Cancer. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 9, Page 262-267, Year 2018 |
Publish date | Dec 28, 2017 (structure data deposition date) |
Authors | Xiang, Q. / Zhang, Y. / Li, J. / Xue, X. / Wang, C. / Song, M. / Zhang, C. / Wang, R. / Li, C. / Wu, C. ...Xiang, Q. / Zhang, Y. / Li, J. / Xue, X. / Wang, C. / Song, M. / Zhang, C. / Wang, R. / Li, C. / Wu, C. / Zhou, Y. / Yang, X. / Li, G. / Ding, K. / Xu, Y. |
External links | Acs Med. Chem. Lett. / PubMed:29541371 |
Methods | X-ray diffraction |
Resolution | 1.42 - 1.62 Å |
Structure data | PDB-5z1r: PDB-5z1s: PDB-5z1t: |
Chemicals | ChemComp-EFL: ChemComp-EDO: ChemComp-GOL: ChemComp-NO3: ChemComp-HOH: ChemComp-EFM: ChemComp-EFN: |
Source |
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Keywords | TRANSCRIPTION / BRD4(1) / Bromodomain |