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-Structure paper
Title | Pharmacological and Structural Characterizations of Naquotinib, a Novel Third-Generation EGFR Tyrosine Kinase Inhibitor, inEGFR-Mutated Non-Small Cell Lung Cancer. |
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Journal, issue, pages | Mol. Cancer Ther., Vol. 17, Page 740-750, Year 2018 |
Publish date | Aug 28, 2017 (structure data deposition date) |
Authors | Hirano, T. / Yasuda, H. / Hamamoto, J. / Nukaga, S. / Masuzawa, K. / Kawada, I. / Naoki, K. / Niimi, T. / Mimasu, S. / Sakagami, H. ...Hirano, T. / Yasuda, H. / Hamamoto, J. / Nukaga, S. / Masuzawa, K. / Kawada, I. / Naoki, K. / Niimi, T. / Mimasu, S. / Sakagami, H. / Soejima, K. / Betsuyaku, T. |
External links | Mol. Cancer Ther. / PubMed:29467275 |
Methods | X-ray diffraction |
Resolution | 3.25 Å |
Structure data | PDB-5y9t: |
Chemicals | ChemComp-8RC: |
Source |
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Keywords | TRANSFERASE / Kinase |