+Search query
-Structure paper
Title | Fragment-Based Discovery of Pyrimido[1,2-b]indazole PDE10A Inhibitors. |
---|---|
Journal, issue, pages | Chem. Pharm. Bull., Vol. 66, Page 286-294, Year 2018 |
Publish date | Jun 23, 2017 (structure data deposition date) |
![]() | Chino, A. / Seo, R. / Amano, Y. / Namatame, I. / Hamaguchi, W. / Honbou, K. / Mihara, T. / Yamazaki, M. / Tomishima, M. / Masuda, N. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.44 - 2.77 Å |
Structure data | ![]() PDB-5xui: ![]() PDB-5xuj: |
Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-MG: ![]() ChemComp-8G3: ![]() ChemComp-HOH: ![]() ChemComp-8G6: |
Source |
|
![]() | HYDROLASE/HYDROLASE INHIBITOR / PDE10A inhibitor / HYDROLASE / HYDROLASE-HYDROLASE INHIBITOR complex |