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Title | Structure-based design, synthesis, and biological evaluation of imidazo[1,2-b]pyridazine-based p38 MAP kinase inhibitors. |
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Journal, issue, pages | Bioorg. Med. Chem., Vol. 26, Page 647-660, Year 2018 |
Publish date | Jul 23, 2017 (structure data deposition date) |
![]() | Kaieda, A. / Takahashi, M. / Takai, T. / Goto, M. / Miyazaki, T. / Hori, Y. / Unno, S. / Kawamoto, T. / Tanaka, T. / Itono, S. ...Kaieda, A. / Takahashi, M. / Takai, T. / Goto, M. / Miyazaki, T. / Hori, Y. / Unno, S. / Kawamoto, T. / Tanaka, T. / Itono, S. / Takagi, T. / Hamada, T. / Shirasaki, M. / Okada, K. / Snell, G. / Bragstad, K. / Sang, B.C. / Uchikawa, O. / Miwatashi, S. |
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Methods | X-ray diffraction |
Resolution | 1.6 - 2 Å |
Structure data | ![]() PDB-5wjj: ![]() PDB-6anl: |
Chemicals | ![]() ChemComp-AQY: ![]() ChemComp-HOH: ![]() ChemComp-T75: |
Source |
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![]() | Transferase/Transferase Inhibitor / Transferase-Transferase Inhibitor complex / TRANSFERASE |