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-Structure paper
Title | Takinib, a Selective TAK1 Inhibitor, Broadens the Therapeutic Efficacy of TNF-alpha Inhibition for Cancer and Autoimmune Disease. |
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Journal, issue, pages | Cell Chem Biol, Vol. 24, Page 1029-1039.e7, Year 2017 |
Publish date | Mar 14, 2017 (structure data deposition date) |
Authors | Totzke, J. / Gurbani, D. / Raphemot, R. / Hughes, P.F. / Bodoor, K. / Carlson, D.A. / Loiselle, D.R. / Bera, A.K. / Eibschutz, L.S. / Perkins, M.M. ...Totzke, J. / Gurbani, D. / Raphemot, R. / Hughes, P.F. / Bodoor, K. / Carlson, D.A. / Loiselle, D.R. / Bera, A.K. / Eibschutz, L.S. / Perkins, M.M. / Eubanks, A.L. / Campbell, P.L. / Fox, D.A. / Westover, K.D. / Haystead, T.A.J. / Derbyshire, E.R. |
External links | Cell Chem Biol / PubMed:28820959 |
Methods | X-ray diffraction |
Resolution | 2.006 Å |
Structure data | PDB-5v5n: |
Chemicals | ChemComp-EDH: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE inhibitor / TAK1 / inhibitor / hydrogen bond / DFG-in / TRANSFERASE-TRANSFERASE inhibitor complex |