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-Structure paper
Title | Structure of a Myeloid cell leukemia-1 (Mcl-1) inhibitor bound to drug site 3 of Human Serum Albumin. |
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Journal, issue, pages | Bioorg. Med. Chem., Vol. 25, Page 3087-3092, Year 2017 |
Publish date | Jan 17, 2017 (structure data deposition date) |
![]() | Zhao, B. / Sensintaffar, J. / Bian, Z. / Belmar, J. / Lee, T. / Olejniczak, E.T. / Fesik, S.W. |
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Methods | X-ray diffraction |
Resolution | 2.7 Å |
Structure data | ![]() PDB-5ujb: |
Chemicals | ![]() ChemComp-6AK: ![]() ChemComp-PO4: |
Source |
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![]() | TRANSPORT PROTEIN / Human Serum Albumin / Free fraction / Apoptosis / cancer / Mcl-1 / drug discovery |