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-Structure paper
Title | X-ray crystal structure of plasmin with tranexamic acid-derived active site inhibitors. |
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Journal, issue, pages | Blood Adv, Vol. 1, Page 766-771, Year 2017 |
Publish date | Jan 8, 2017 (structure data deposition date) |
![]() | Law, R.H.P. / Wu, G. / Leung, E.W.W. / Hidaka, K. / Quek, A.J. / Caradoc-Davies, T.T. / Jeevarajah, D. / Conroy, P.J. / Kirby, N.M. / Norton, R.S. ...Law, R.H.P. / Wu, G. / Leung, E.W.W. / Hidaka, K. / Quek, A.J. / Caradoc-Davies, T.T. / Jeevarajah, D. / Conroy, P.J. / Kirby, N.M. / Norton, R.S. / Tsuda, Y. / Whisstock, J.C. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.2 - 1.38 Å |
Structure data | ![]() PDB-5ugd: ![]() PDB-5ugg: |
Chemicals | ![]() ChemComp-89S: ![]() ChemComp-HOH: ![]() ChemComp-89M: |
Source |
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![]() | HYDROLASE/INHIBITOR / Fibrinolysis / YO / Plasmin / Inhibitor / HYDROLASE-INHIBITOR complex |