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-Structure paper
Title | Discovery of a First-in-Class Receptor Interacting Protein 1 (RIP1) Kinase Specific Clinical Candidate (GSK2982772) for the Treatment of Inflammatory Diseases. |
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Journal, issue, pages | J. Med. Chem., Vol. 60, Page 1247-1261, Year 2017 |
Publish date | Nov 15, 2016 (structure data deposition date) |
Authors | Harris, P.A. / Berger, S.B. / Jeong, J.U. / Nagilla, R. / Bandyopadhyay, D. / Campobasso, N. / Capriotti, C.A. / Cox, J.A. / Dare, L. / Dong, X. ...Harris, P.A. / Berger, S.B. / Jeong, J.U. / Nagilla, R. / Bandyopadhyay, D. / Campobasso, N. / Capriotti, C.A. / Cox, J.A. / Dare, L. / Dong, X. / Eidam, P.M. / Finger, J.N. / Hoffman, S.J. / Kang, J. / Kasparcova, V. / King, B.W. / Lehr, R. / Lan, Y. / Leister, L.K. / Lich, J.D. / MacDonald, T.T. / Miller, N.A. / Ouellette, M.T. / Pao, C.S. / Rahman, A. / Reilly, M.A. / Rendina, A.R. / Rivera, E.J. / Schaeffer, M.C. / Sehon, C.A. / Singhaus, R.R. / Sun, H.H. / Swift, B.A. / Totoritis, R.D. / Vossenkamper, A. / Ward, P. / Wisnoski, D.D. / Zhang, D. / Marquis, R.W. / Gough, P.J. / Bertin, J. |
External links | J. Med. Chem. / PubMed:28151659 |
Methods | X-ray diffraction |
Resolution | 2.56 Å |
Structure data | PDB-5tx5: |
Chemicals | ChemComp-7MJ: ChemComp-HOH: |
Source |
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Keywords | transferase/transferase inhibitor / kinase domain Inhibitor necrosis / transferase-transferase inhibitor complex |