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-Structure paper
Title | Potent competitive inhibition of human ribonucleotide reductase by a nonnucleoside small molecule. |
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Journal, issue, pages | Proc. Natl. Acad. Sci. U.S.A., Vol. 114, Page 8241-8246, Year 2017 |
Publish date | Nov 7, 2016 (structure data deposition date) |
![]() | Ahmad, M.F. / Alam, I. / Huff, S.E. / Pink, J. / Flanagan, S.A. / Shewach, D. / Misko, T.A. / Oleinick, N.L. / Harte, W.E. / Viswanathan, R. ...Ahmad, M.F. / Alam, I. / Huff, S.E. / Pink, J. / Flanagan, S.A. / Shewach, D. / Misko, T.A. / Oleinick, N.L. / Harte, W.E. / Viswanathan, R. / Harris, M.E. / Dealwis, C.G. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.66 Å |
Structure data | ![]() PDB-5tus: |
Chemicals | ![]() ChemComp-TTP: ![]() ChemComp-MG: ![]() ChemComp-7LL: ![]() ChemComp-HOH: |
Source |
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![]() | OXIDOREDUCTASE / Ribonucleotide Reductase / small molecule inhibitor / active site inhibitor / competitive inhibitor |