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-Structure paper
Title | SAR405838: an optimized inhibitor of MDM2-p53 interaction that induces complete and durable tumor regression. |
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Journal, issue, pages | Cancer Res., Vol. 74, Page 5855-5865, Year 2014 |
Publish date | Oct 26, 2016 (structure data deposition date) |
Authors | Wang, S. / Sun, W. / Zhao, Y. / McEachern, D. / Meaux, I. / Barriere, C. / Stuckey, J.A. / Meagher, J.L. / Bai, L. / Liu, L. ...Wang, S. / Sun, W. / Zhao, Y. / McEachern, D. / Meaux, I. / Barriere, C. / Stuckey, J.A. / Meagher, J.L. / Bai, L. / Liu, L. / Hoffman-Luca, C.G. / Lu, J. / Shangary, S. / Yu, S. / Bernard, D. / Aguilar, A. / Dos-Santos, O. / Besret, L. / Guerif, S. / Pannier, P. / Gorge-Bernat, D. / Debussche, L. |
External links | Cancer Res. / PubMed:25145672 |
Methods | X-ray diffraction |
Resolution | 2.1 Å |
Structure data | PDB-5trf: |
Chemicals | ChemComp-7HC: ChemComp-SO4: ChemComp-GOL: ChemComp-HOH: |
Source |
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Keywords | LIGASE/LIGASE INHIBITOR / P53-BINDING PROTEIN / ONCOPROTEIN / DOUBLE MINUTE 2 PROTEIN / SMALL MOLECULE INHIBITOR / LIGASE-LIGASE INHIBITOR complex |