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-Structure paper
Title | Buried Hydrogen Bond Interactions Contribute to the High Potency of Complement Factor D Inhibitors. |
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Journal, issue, pages | ACS Med Chem Lett, Vol. 7, Page 1092-1096, Year 2016 |
Publish date | Sep 14, 2016 (structure data deposition date) |
Authors | Yang, C.Y. / Phillips, J.G. / Stuckey, J.A. / Bai, L. / Sun, H. / Delproposto, J. / Brown, W.C. / Chinnaswamy, K. |
External links | ACS Med Chem Lett / PubMed:27994744 |
Methods | X-ray diffraction |
Resolution | 3.15 - 3.37 Å |
Structure data | PDB-5tca: PDB-5tcc: |
Chemicals | ChemComp-J55: ChemComp-HOH: ChemComp-J56: |
Source |
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Keywords | HYDROLASE/HYDROLASE INHIBITOR / serine protease / inhibitor / HYDROLASE-HYDROLASE INHIBITOR complex |