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-Structure paper
Title | Crystal Structure of the Emerging Cancer Target MTHFD2 in Complex with a Substrate-Based Inhibitor. |
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Journal, issue, pages | Cancer Res., Vol. 77, Page 937-948, Year 2017 |
Publish date | Sep 14, 2016 (structure data deposition date) |
Authors | Gustafsson, R. / Jemth, A.S. / Gustafsson, N.M. / Farnegardh, K. / Loseva, O. / Wiita, E. / Bonagas, N. / Dahllund, L. / Llona-Minguez, S. / Haggblad, M. ...Gustafsson, R. / Jemth, A.S. / Gustafsson, N.M. / Farnegardh, K. / Loseva, O. / Wiita, E. / Bonagas, N. / Dahllund, L. / Llona-Minguez, S. / Haggblad, M. / Henriksson, M. / Andersson, Y. / Homan, E. / Helleday, T. / Stenmark, P. |
External links | Cancer Res. / PubMed:27899380 |
Methods | X-ray diffraction |
Resolution | 1.89 Å |
Structure data | PDB-5tc4: |
Chemicals | ChemComp-NAD: ChemComp-L34: ChemComp-PO4: ChemComp-HOH: |
Source |
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Keywords | OXIDOREDUCTASE / Inhibitor / Folate / Cofactor / Dehydrogenase |