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-Structure paper
Title | A Small-Molecule Antagonist of HIF2 alpha Is Efficacious in Preclinical Models of Renal Cell Carcinoma. |
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Journal, issue, pages | Cancer Res., Vol. 76, Page 5491-5500, Year 2016 |
Publish date | Sep 12, 2016 (structure data deposition date) |
![]() | Wallace, E.M. / Rizzi, J.P. / Han, G. / Wehn, P.M. / Cao, Z. / Du, X. / Cheng, T. / Czerwinski, R.M. / Dixon, D.D. / Goggin, B.S. ...Wallace, E.M. / Rizzi, J.P. / Han, G. / Wehn, P.M. / Cao, Z. / Du, X. / Cheng, T. / Czerwinski, R.M. / Dixon, D.D. / Goggin, B.S. / Grina, J.A. / Halfmann, M.M. / Maddie, M.A. / Olive, S.R. / Schlachter, S.T. / Tan, H. / Wang, B. / Wang, K. / Xie, S. / Xu, R. / Yang, H. / Josey, J.A. |
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Methods | X-ray diffraction |
Resolution | 1.85 Å |
Structure data | ![]() PDB-5tbm: |
Chemicals | ![]() ChemComp-79A: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSCRIPTION / HIF2 inhibitor HIF2 ligand PAS-B hypoxia inducible factor 2 EPAS1 |