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-Structure paper
Title | Maytansinol Derivatives: Side Reactions as a Chance for New Tubulin Binders. |
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Journal, issue, pages | Chemistry, Vol. 28, Page e202103520-e202103520, Year 2022 |
Publish date | Jul 20, 2021 (structure data deposition date) |
![]() | Marzullo, P. / Boiarska, Z. / Perez-Pena, H. / Abel, A.C. / Alvarez-Bernad, B. / Lucena-Agell, D. / Vasile, F. / Sironi, M. / Altmann, K.H. / Prota, A.E. ...Marzullo, P. / Boiarska, Z. / Perez-Pena, H. / Abel, A.C. / Alvarez-Bernad, B. / Lucena-Agell, D. / Vasile, F. / Sironi, M. / Altmann, K.H. / Prota, A.E. / Diaz, J.F. / Pieraccini, S. / Passarella, D. |
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Methods | X-ray diffraction |
Resolution | 2.25 - 2.75 Å |
Structure data | ![]() PDB-5sb8: ![]() PDB-5sb9: ![]() PDB-5sba: ![]() PDB-5sbb: ![]() PDB-5sbc: ![]() PDB-5sbd: ![]() PDB-5sbe: |
Chemicals | ![]() ChemComp-GTP: ![]() ChemComp-MG: ![]() ChemComp-CA: ![]() ChemComp-GDP: ![]() ChemComp-MES: ![]() ChemComp-IMD: ![]() ChemComp-5IS: ![]() ChemComp-ACP: ![]() ChemComp-HOH: ![]() ChemComp-5IX: ![]() ChemComp-GOL: ![]() ChemComp-5IJ: ![]() ChemComp-5JH: ![]() ChemComp-5JS: ![]() ChemComp-5KI: ![]() ChemComp-5L5: |
Source |
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![]() | CELL CYCLE / TUBULIN FOLD / CYTOSKELETON / MICROTUBULE |