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-Structure paper
Title | Dimethyl fumarate is an allosteric covalent inhibitor of the p90 ribosomal S6 kinases. |
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Journal, issue, pages | Nat Commun, Vol. 9, Page 4344-4344, Year 2018 |
Publish date | May 19, 2017 (structure data deposition date) |
![]() | Andersen, J.L. / Gesser, B. / Funder, E.D. / Nielsen, C.J.F. / Gotfred-Rasmussen, H. / Rasmussen, M.K. / Toth, R. / Gothelf, K.V. / Arthur, J.S.C. / Iversen, L. / Nissen, P. |
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Methods | X-ray diffraction |
Resolution | 1.9 Å |
Structure data | ![]() PDB-5o1s: |
Chemicals | ![]() ChemComp-NA: ![]() ChemComp-9HB: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE / Covalent / Inhibitor / Kinase / allosteric |