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TitleIdentification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs.
Journal, issue, pagesChemMedChem, Vol. 12, Page 1542-1554, Year 2017
Publish dateMar 17, 2017 (structure data deposition date)
AuthorsPirali, T. / Ciraolo, E. / Aprile, S. / Massarotti, A. / Berndt, A. / Griglio, A. / Serafini, M. / Mercalli, V. / Landoni, C. / Campa, C.C. ...Pirali, T. / Ciraolo, E. / Aprile, S. / Massarotti, A. / Berndt, A. / Griglio, A. / Serafini, M. / Mercalli, V. / Landoni, C. / Campa, C.C. / Margaria, J.P. / Silva, R.L. / Grosa, G. / Sorba, G. / Williams, R. / Hirsch, E. / Tron, G.C.
External linksChemMedChem / PubMed:28857471
MethodsX-ray diffraction
Resolution2.9 Å
Structure data

PDB-5ngb:
X-Ray Diffraction Crystal Structure of the murine PI3K p110delta in complex with a pan inhibitor
Method: X-RAY DIFFRACTION / Resolution: 2.9 Å

Chemicals

ChemComp-8WH:
3-[[4-(2-morpholin-4-yl-4-oxidanylidene-3~{H}-quinolin-8-yl)-1,2,3-triazol-1-yl]methyl]benzoic acid

Source
  • mus musculus (house mouse)
KeywordsTRANSFERASE / PI3K p110

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