+Search query
-Structure paper
Title | Discovery of New Bromodomain Scaffolds by Biosensor Fragment Screening. |
---|---|
Journal, issue, pages | ACS Med Chem Lett, Vol. 7, Page 1213-1218, Year 2016 |
Publish date | Sep 11, 2016 (structure data deposition date) |
![]() | Navratilova, I. / Aristotelous, T. / Picaud, S. / Chaikuad, A. / Knapp, S. / Filappakopoulos, P. / Hopkins, A.L. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.61 - 2.05 Å |
Structure data | ![]() PDB-5luu: ![]() PDB-5lvq: ![]() PDB-5lvr: ![]() PDB-5tb6: |
Chemicals | ![]() ChemComp-EDO: ![]() ChemComp-77X: ![]() ChemComp-HOH: ![]() ChemComp-2LX: ![]() ChemComp-DMS: ![]() ChemComp-78Y: |
Source |
|
![]() | TRANSCRIPTION / Fragment / complex / bromodomain / Structural Genomics / Structural Genomics Consortium / SGC / TRANSFERASE / SIGNALING PROTEIN / HISTONE ACETYLTRANSFERASE KAT2B / HISTONE / ACETYLATION / ACETYLLYSINE / EPIGENETICS / STRUCTURAL GENOMICS CONSORTIUM (SGC) / trasnferase |