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-Structure paper
Title | Evolution of a Novel, Orally Bioavailable Series of PI3K delta Inhibitors from an Inhaled Lead for the Treatment of Respiratory Disease. |
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Journal, issue, pages | J. Med. Chem., Vol. 59, Page 7239-7251, Year 2016 |
Publish date | Jun 1, 2016 (structure data deposition date) |
Authors | Amour, A. / Barton, N. / Cooper, A.W. / Inglis, G. / Jamieson, C. / Luscombe, C.N. / Morrell, J. / Peace, S. / Perez, D. / Rowland, P. ...Amour, A. / Barton, N. / Cooper, A.W. / Inglis, G. / Jamieson, C. / Luscombe, C.N. / Morrell, J. / Peace, S. / Perez, D. / Rowland, P. / Tame, C. / Uddin, S. / Vitulli, G. / Wellaway, N. |
External links | J. Med. Chem. / PubMed:27429068 |
Methods | X-ray diffraction |
Resolution | 3.06 Å |
Structure data | PDB-5l72: |
Chemicals | ChemComp-6PF: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / PI3 kinase delta |