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-Structure paper
Title | Development of Specific, Irreversible Inhibitors for a Receptor Tyrosine Kinase EphB3. |
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Journal, issue, pages | J. Am. Chem. Soc., Vol. 138, Page 10554-10560, Year 2016 |
Publish date | May 30, 2016 (structure data deposition date) |
![]() | Kung, A. / Chen, Y.C. / Schimpl, M. / Ni, F. / Zhu, J. / Turner, M. / Molina, H. / Overman, R. / Zhang, C. |
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Methods | X-ray diffraction |
Resolution | 1.88 - 2.26 Å |
Structure data | ![]() PDB-5l6o: ![]() PDB-5l6p: |
Chemicals | ![]() ChemComp-6P6: ![]() ChemComp-DIO: ![]() ChemComp-HOH: ![]() ChemComp-6P8: |
Source |
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![]() | TRANSFERASE / Kinase / Irreversible Inhibitor / Quinazoline / Signaling |