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Structure paper

TitleIdentification of potent, selective KDM5 inhibitors.
Journal, issue, pagesBioorg. Med. Chem. Lett., Vol. 26, Page 4350-4354, Year 2016
Publish dateJul 7, 2016 (structure data deposition date)
AuthorsGehling, V.S. / Bellon, S.F. / Harmange, J.C. / LeBlanc, Y. / Poy, F. / Odate, S. / Buker, S. / Lan, F. / Arora, S. / Williamson, K.E. ...Gehling, V.S. / Bellon, S.F. / Harmange, J.C. / LeBlanc, Y. / Poy, F. / Odate, S. / Buker, S. / Lan, F. / Arora, S. / Williamson, K.E. / Sandy, P. / Cummings, R.T. / Bailey, C.M. / Bergeron, L. / Mao, W. / Gustafson, A. / Liu, Y. / VanderPorten, E. / Audia, J.E. / Trojer, P. / Albrecht, B.K.
External linksBioorg. Med. Chem. Lett. / PubMed:27476424
MethodsX-ray diffraction
Resolution1.9 Å
Structure data

PDB-5kr7:
KDM4C bound to pyrazolo-pyrimidine scaffold
Method: X-RAY DIFFRACTION / Resolution: 1.9 Å

Chemicals

ChemComp-FE2:
Unknown entry

ChemComp-ZN:
Unknown entry

ChemComp-6X9:
6-ethyl-2,5-dimethyl-7-oxidanylidene-4~{H}-pyrazolo[1,5-a]pyrimidine-3-carbonitrile

ChemComp-CL:
Unknown entry

ChemComp-HOH:
WATER

Source
  • homo sapiens (human)
KeywordsOXIDOREDUCTASE / inhibitor / histone / lysine demethylase

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