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-Structure paper
Title | Assessment of Bromodomain Target Engagement by a Series of BI2536 Analogues with Miniaturized BET-BRET. |
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Journal, issue, pages | ChemMedChem, Vol. 11, Page 2575-2581, Year 2016 |
Publish date | Jun 17, 2016 (structure data deposition date) |
Authors | Koblan, L.W. / Buckley, D.L. / Ott, C.J. / Fitzgerald, M.E. / Ember, S.W. / Zhu, J.Y. / Liu, S. / Roberts, J.M. / Remillard, D. / Vittori, S. ...Koblan, L.W. / Buckley, D.L. / Ott, C.J. / Fitzgerald, M.E. / Ember, S.W. / Zhu, J.Y. / Liu, S. / Roberts, J.M. / Remillard, D. / Vittori, S. / Zhang, W. / Schonbrunn, E. / Bradner, J.E. |
External links | ChemMedChem / PubMed:27862999 |
Methods | X-ray diffraction |
Resolution | 1.51 Å |
Structure data | PDB-5kj0: |
Chemicals | ChemComp-6TB: ChemComp-EDO: ChemComp-HOH: |
Source |
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Keywords | TRANSCRIPTION/INHIBITOR / BROMODOMAIN / CAP / HUNK1 / MCAP / PROTEIN BINDING-INHIBITOR COMPLEX / MITOTIC CHROMOSOME ASSOCIATED PROTEIN / CELL CYCLE / INHIBITOR / TRANSCRIPTION-INHIBITOR COMPLEX |