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-Structure paper
Title | SETDB1 in complex with an early stage, low affinity fragment candidate modelled at reduced occupancy |
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Journal, issue, pages | To Be Published |
Publish date | Jun 6, 2016 (structure data deposition date) |
Authors | Tempel, W. / Harding, R.J. / Mader, P. / Dobrovetsky, E. / Walker, J.R. / Brown, P.J. / Schapira, M. / Arrowsmith, C.H. / Edwards, A.M. / Santhakumar, S. / Structural Genomics Consortium (SGC) |
External links | Search PubMed |
Methods | X-ray diffraction |
Resolution | 1.47 - 1.7 Å |
Structure data | PDB-5kch: PDB-5kco: |
Chemicals | ChemComp-UNX: ChemComp-DMS: ChemComp-SO4: ChemComp-6RN: ChemComp-HOH: ChemComp-6RO: |
Source |
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Keywords | TRANSFERASE / Fragment Screening / DIAMOND I04-1 XCHEM / PANDDA / Structural Genomics / Structural Genomics Consortium / SGC |