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-Structure paper
Title | Development of ML390: A Human DHODH Inhibitor That Induces Differentiation in Acute Myeloid Leukemia. |
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Journal, issue, pages | ACS Med Chem Lett, Vol. 7, Page 1112-1117, Year 2016 |
Publish date | May 31, 2016 (structure data deposition date) |
Authors | Lewis, T.A. / Sykes, D.B. / Law, J.M. / Munoz, B. / Rustiguel, J.K. / Nonato, M.C. / Scadden, D.T. / Schreiber, S.L. |
External links | ACS Med Chem Lett / PubMed:27994748 |
Methods | X-ray diffraction |
Resolution | 1.66 - 1.7 Å |
Structure data | PDB-5k9c: PDB-5k9d: |
Chemicals | ChemComp-FNR: ChemComp-ORO: ChemComp-MLJ: ChemComp-SO4: ChemComp-ACT: ChemComp-CL: ChemComp-GOL: ChemComp-HOH: ChemComp-CE9: |
Source |
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Keywords | OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR / Oxidoreductase / alpha/beta barrel / inhibitor / OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR complex |