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-Structure paper
Title | Discovery of Novel, Orally Bioavailable beta-Amino Acid Azaindole Inhibitors of Influenza PB2. |
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Journal, issue, pages | ACS Med Chem Lett, Vol. 8, Page 256-260, Year 2017 |
Publish date | May 10, 2016 (structure data deposition date) |
Authors | Farmer, L.J. / Clark, M.P. / Boyd, M.J. / Perola, E. / Jones, S.M. / Tsai, A. / Jacobs, M.D. / Bandarage, U.K. / Ledeboer, M.W. / Wang, T. ...Farmer, L.J. / Clark, M.P. / Boyd, M.J. / Perola, E. / Jones, S.M. / Tsai, A. / Jacobs, M.D. / Bandarage, U.K. / Ledeboer, M.W. / Wang, T. / Deng, H. / Ledford, B. / Gu, W. / Duffy, J.P. / Bethiel, R.S. / Shannon, D. / Byrn, R.A. / Leeman, J.R. / Rijnbrand, R. / Bennett, H.B. / O'Brien, C. / Memmott, C. / Nti-Addae, K. / Bennani, Y.L. / Charifson, P.S. |
External links | ACS Med Chem Lett / PubMed:28197322 |
Methods | X-ray diffraction |
Resolution | 2.69 - 2.93 Å |
Structure data | PDB-5jun: PDB-5jur: |
Chemicals | ChemComp-6NU: ChemComp-HOH: ChemComp-6NS: |
Source |
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Keywords | RNA BINDING PROTEIN / flu / polymerase / nucleotide binding / inhibitor |