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-Structure paper
Title | Inhibitor Selectivity for Cyclin-Dependent Kinase 7: A Structural, Thermodynamic, and Modelling Study. |
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Journal, issue, pages | ChemMedChem, Vol. 12, Page 372-380, Year 2017 |
Publish date | May 4, 2016 (structure data deposition date) |
![]() | Hazel, P. / Kroll, S.H. / Bondke, A. / Barbazanges, M. / Patel, H. / Fuchter, M.J. / Coombes, R.C. / Ali, S. / Barrett, A.G. / Freemont, P.S. |
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Methods | X-ray diffraction |
Resolution | 1.94 Å |
Structure data | ![]() PDB-5jq5: ![]() PDB-5jq8: |
Chemicals | ![]() ChemComp-ACT: ![]() ChemComp-I74: ![]() ChemComp-HOH: ![]() ChemComp-I73: |
Source |
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![]() | transferase/transferase inhibitor / CDK2 / kinase / inhibitor / transferase-transferase inhibitor complex / Kinase inhibitor |