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-Structure paper
Title | Pyrazolylamine Derivatives Reveal the Conformational Switching between Type I and Type II Binding Modes of Anaplastic Lymphoma Kinase (ALK). |
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Journal, issue, pages | J. Med. Chem., Vol. 59, Page 3906-3919, Year 2016 |
Publish date | Mar 18, 2016 (structure data deposition date) |
Authors | Tu, C.H. / Lin, W.H. / Peng, Y.H. / Hsu, T. / Wu, J.S. / Chang, C.Y. / Lu, C.T. / Lyu, P.C. / Shih, C. / Jiaang, W.T. / Wu, S.Y. |
External links | J. Med. Chem. / PubMed:27031565 |
Methods | X-ray diffraction |
Resolution | 1.88 - 2.1 Å |
Structure data | PDB-5iug: PDB-5iuh: PDB-5iui: |
Chemicals | ChemComp-729: ChemComp-HOH: ChemComp-34Y: ChemComp-45Q: |
Source |
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Keywords | TRANSFERASE / CATALYTIC DOMAIN |