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-Structure paper
| Title | Design and Development of a Series of Potent and Selective Type II Inhibitors of CDK8. |
|---|---|
| Journal, issue, pages | Acs Med. Chem. Lett., Vol. 7, Page 595-600, Year 2016 |
| Publish date | Jan 28, 2016 (structure data deposition date) |
Authors | Bergeron, P. / Koehler, M.F. / Blackwood, E.M. / Bowman, K. / Clark, K. / Firestein, R. / Kiefer, J.R. / Maskos, K. / McCleland, M.L. / Orren, L. ...Bergeron, P. / Koehler, M.F. / Blackwood, E.M. / Bowman, K. / Clark, K. / Firestein, R. / Kiefer, J.R. / Maskos, K. / McCleland, M.L. / Orren, L. / Ramaswamy, S. / Salphati, L. / Schmidt, S. / Schneider, E.V. / Wu, J. / Beresini, M. |
External links | Acs Med. Chem. Lett. / PubMed:27326333 |
| Methods | X-ray diffraction |
| Resolution | 2.39 Å |
| Structure data | ![]() PDB-5hvy: |
| Chemicals | ![]() ChemComp-66X: ![]() ChemComp-FMT: ![]() ChemComp-CL: ![]() ChemComp-HOH: |
| Source |
|
Keywords | Transferase/Transcription / Transferase-Transcription complex |
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homo sapiens (human)
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