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Title | Identification and in Vivo Evaluation of Liver X Receptor beta-Selective Agonists for the Potential Treatment of Alzheimer's Disease. |
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Journal, issue, pages | J. Med. Chem., Vol. 59, Page 3489-3498, Year 2016 |
Publish date | Jan 13, 2016 (structure data deposition date) |
Authors | Stachel, S.J. / Zerbinatti, C. / Rudd, M.T. / Cosden, M. / Suon, S. / Nanda, K.K. / Wessner, K. / DiMuzio, J. / Maxwell, J. / Wu, Z. ...Stachel, S.J. / Zerbinatti, C. / Rudd, M.T. / Cosden, M. / Suon, S. / Nanda, K.K. / Wessner, K. / DiMuzio, J. / Maxwell, J. / Wu, Z. / Uslaner, J.M. / Michener, M.S. / Szczerba, P. / Brnardic, E. / Rada, V. / Kim, Y. / Meissner, R. / Wuelfing, P. / Yuan, Y. / Ballard, J. / Holahan, M. / Klein, D.J. / Lu, J. / Fradera, X. / Parthasarathy, G. / Uebele, V.N. / Chen, Z. / Li, Y. / Li, J. / Cooke, A.J. / Bennett, D.J. / Bilodeau, M.T. / Renger, J. |
External links | J. Med. Chem. / PubMed:27011007 |
Methods | X-ray diffraction |
Resolution | 1.72 - 2.6 Å |
Structure data | PDB-5hjp: PDB-5hjs: |
Chemicals | ChemComp-668: ChemComp-PEG: ChemComp-HOH: ChemComp-SO4: |
Source |
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Keywords | SIGNALING PROTEIN / Agonist / Alzheimer's |