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-Structure paper
Title | Potent and Selective CK2 Kinase Inhibitors with Effects on Wnt Pathway Signaling in Vivo. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 7, Page 300-305, Year 2016 |
Publish date | Dec 23, 2015 (structure data deposition date) |
![]() | Dowling, J.E. / Alimzhanov, M. / Bao, L. / Chuaqui, C. / Denz, C.R. / Jenkins, E. / Larsen, N.A. / Lyne, P.D. / Pontz, T. / Ye, Q. ...Dowling, J.E. / Alimzhanov, M. / Bao, L. / Chuaqui, C. / Denz, C.R. / Jenkins, E. / Larsen, N.A. / Lyne, P.D. / Pontz, T. / Ye, Q. / Holdgate, G.A. / Snow, L. / O'Connell, N. / Ferguson, A.D. |
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Methods | X-ray diffraction |
Resolution | 2 - 2.55 Å |
Structure data | ![]() PDB-5h8b: ![]() PDB-5h8e: ![]() PDB-5h8g: |
Chemicals | ![]() ChemComp-SO4: ![]() ChemComp-EDO: ![]() ChemComp-5Y2: ![]() ChemComp-HOH: ![]() ChemComp-5Y3: ![]() ChemComp-CL: ![]() ChemComp-5Y4: |
Source |
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![]() | Transferase/Transferase Inhibitor / Kinase / Inhibitor / CK2 / Transferase-Transferase Inhibitor complex |