Database of articles cited by EMDB/PDB/SASBDB data

Keywords
Structure methods	All X-ray diffraction NMR electron microscopy small angle scattering neutron diffraction fiber diffraction powder diffraction infrared spectroscopy EPR fluorescence transfer theoretical model Hybrid
Author
Journal
IF	>30 >20 >10 >5 all

Title	Gsk6853, a Chemical Probe for Inhibition of the Brpf1 Bromodomain.
Journal, issue, pages	Acs Med. Chem. Lett., Vol. 7, Page 552-, Year 2016
Publish date	May 16, 2016 (structure data deposition date)
Authors	Bamborough, P. / Barnett, H.A. / Becher, I. / Bird, M.J. / Chung, C. / Craggs, P.D. / Demont, E.H. / Diallo, H. / Fallon, D.J. / Gordon, L.J. ...Bamborough, P. / Barnett, H.A. / Becher, I. / Bird, M.J. / Chung, C. / Craggs, P.D. / Demont, E.H. / Diallo, H. / Fallon, D.J. / Gordon, L.J. / Grandi, P. / Hobbs, C.I. / Hooper-Greenhill, E. / Jones, E.J. / Law, R.P. / Le Gall, A. / Lugo, D. / Michon, A. / Mitchell, D.J. / Prinjha, R.K. / Sheppard, R.J. / Watson, A.J.B. / Watson, R.J.
External links	Acs Med. Chem. Lett. / PubMed:27326325
Methods	X-ray diffraction
Resolution	1.6 - 1.96 Å
Structure data	PDB-5g4r: BROMODOMAIN OF HUMAN BRPF1 WITH N-1,3-dimethyl-6-2R-2- methylpiperazin-1-yl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl-2- methoxybenzamide Method: X-RAY DIFFRACTION / Resolution: 1.96 Å PDB-5g4s: BROMODOMAIN OF HUMAN BRPF1 WITH N-1,3-dimethyl-6-2R-2- methylpiperazin-1-yl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl-N- ethyl-2-methoxybenzamide Method: X-RAY DIFFRACTION / Resolution: 1.6 Å
Chemicals	ChemComp-LF1: N-[1,3-dimethyl-6-[(2R)-2-methylpiperazin-1-yl]-2-oxidanylidene-benzimidazol-5-yl]-2-methoxy-benzamide ChemComp-HOH: WATER ChemComp-8VI: N-[1,3-dimethyl-6-[(2R)-2-methylpiperazin-1-yl]-2-oxidanylidene-benzimidazol-5-yl]-N-ethyl-2-methoxy-benzamide ChemComp-EDO: 1,2-ETHANEDIOL
Source	homo sapiens (human)
Keywords	TRANSCRIPTION