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-Structure paper
Title | Cryptosporidium and Toxoplasma Parasites are Inhibited by a Benzoxaborole Targeting Leucyl-tRNA Synthetase. |
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Journal, issue, pages | Antimicrob. Agents Chemother., Vol. 60, Page 5817-, Year 2016 |
Publish date | Nov 20, 2015 (structure data deposition date) |
![]() | Palencia, A. / Liu, R. / Lukarska, M. / Gut, J. / Bougdour, A. / Touquet, B. / Wang, E. / Li, X. / Alley, M.R.K. / Freund, Y.R. ...Palencia, A. / Liu, R. / Lukarska, M. / Gut, J. / Bougdour, A. / Touquet, B. / Wang, E. / Li, X. / Alley, M.R.K. / Freund, Y.R. / Rosenthal, P.J. / Hakimi, M. / Cusack, S. |
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Methods | X-ray diffraction |
Resolution | 1.77 - 2.7 Å |
Structure data | ![]() PDB-5fog: ![]() PDB-5fol: ![]() PDB-5fom: ![]() PDB-5fon: |
Chemicals | ![]() ChemComp-VRT: ![]() ChemComp-EDO: ![]() ChemComp-K: ![]() ChemComp-HOH: ![]() ChemComp-PO4: ![]() ChemComp-SO8: ![]() ChemComp-A2H: |
Source |
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![]() | LYASE / CRYPTOSPORIDIUM / LEUCINE-TRNA LIGASE (LEURS) ACTIVITY / ATP + L-LEUCINE + TRNA(LEUCINE) GIVE AMP + DIPHOSPHATE + L-LEUCYL-TRNA(LEUCINE) / POST-TRANSFER EDITING ACTIVITY OF LEURS / AMINOACYL-TRNA SYNTHETASE / PROTEIN BIOSYNTHESIS / NOVEL BORON INHIBITORS OF THE EDITING SITE OF LEURS / LIGASE |