+Search query
-Structure paper
Title | Exploring Selective Inhibition of the First Bromodomain of the Human Bromodomain and Extra-terminal Domain (BET) Proteins. |
---|---|
Journal, issue, pages | J. Med. Chem., Vol. 59, Page 1634-1641, Year 2016 |
Publish date | Oct 27, 2015 (structure data deposition date) |
Authors | Raux, B. / Voitovich, Y. / Derviaux, C. / Lugari, A. / Rebuffet, E. / Milhas, S. / Priet, S. / Roux, T. / Trinquet, E. / Guillemot, J.C. ...Raux, B. / Voitovich, Y. / Derviaux, C. / Lugari, A. / Rebuffet, E. / Milhas, S. / Priet, S. / Roux, T. / Trinquet, E. / Guillemot, J.C. / Knapp, S. / Brunel, J.M. / Fedorov, A.Y. / Collette, Y. / Roche, P. / Betzi, S. / Combes, S. / Morelli, X. |
External links | J. Med. Chem. / PubMed:26735842 |
Methods | X-ray diffraction |
Resolution | 1.05 - 2.21 Å |
Structure data | PDB-5egu: PDB-5ei4: PDB-5eis: |
Chemicals | ChemComp-5NQ: ChemComp-EDO: ChemComp-HOH: ChemComp-5NV: ChemComp-5OU: |
Source |
|
Keywords | TRANSCRIPTION / INHIBITOR / HISTONE / EPIGENETIC READER / BROMODOMAIN / BRD4 / Brd4_BD1 / Brd4_BD1 06-NOV / Brd4_BD1 29-O |