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-Structure paper
Title | The "Gatekeeper" Residue Influences the Mode of Binding of Acetyl Indoles to Bromodomains. |
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Journal, issue, pages | J. Med. Chem., Vol. 59, Page 3087-3097, Year 2016 |
Publish date | Aug 14, 2015 (structure data deposition date) |
![]() | Unzue, A. / Zhao, H. / Lolli, G. / Dong, J. / Zhu, J. / Zechner, M. / Dolbois, A. / Caflisch, A. / Nevado, C. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.35 - 1.783 Å |
Structure data | ![]() PDB-5d7x: ![]() PDB-5e73: ![]() PDB-5e74: |
Chemicals | ![]() ChemComp-NO3: ![]() ChemComp-XZ8: ![]() ChemComp-HOH: ![]() ChemComp-UO1: ![]() ChemComp-5KH: |
Source |
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![]() | DNA BINDING PROTEIN / Bromodomain and PHD finger-containing protein 1(BRPF1) / monocytic leukemia zinc-finger (MOZ) / Inhibitor / TRANSCRIPTION / four helical bundle |