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Structure paper

TitleRVX-297- a novel BD2 selective inhibitor of BET bromodomains.
Journal, issue, pagesBiochem. Biophys. Res. Commun., Vol. 477, Page 62-67, Year 2016
Publish dateSep 22, 2015 (structure data deposition date)
AuthorsKharenko, O.A. / Gesner, E.M. / Patel, R.G. / Norek, K. / White, A. / Fontano, E. / Suto, R.K. / Young, P.R. / McLure, K.G. / Hansen, H.C.
External linksBiochem. Biophys. Res. Commun. / PubMed:27282480
MethodsX-ray diffraction
Resolution1.12 - 1.55 Å
Structure data

PDB-5dw1:
X-ray crystal structure of human BRD2(BD2) in complex with RVX297 to 1.55 A resolution
Method: X-RAY DIFFRACTION / Resolution: 1.55 Å

PDB-5dw2:
X-ray crystal structure of human BRD4(BD1) in complex with RVX297 to 1.12 A resolution
Method: X-RAY DIFFRACTION / Resolution: 1.12 Å

Chemicals

ChemComp-5GD:
2-{3,5-dimethyl-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-5,7-dimethoxyquinazolin-4(3H)-one

ChemComp-NA:
Unknown entry

ChemComp-HOH:
WATER

ChemComp-EDO:
1,2-ETHANEDIOL

Source
  • homo sapiens (human)
KeywordsPROTEIN BINDING/INHIBITOR / bromodomain / PROTEIN BINDING-INHIBITOR complex

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