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-Structure paper
Title | Protein-Protein Interaction Inhibition (2P2I)-Oriented Chemical Library Accelerates Hit Discovery. |
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Journal, issue, pages | Acs Chem. Biol., Vol. 11, Page 2140-2148, Year 2016 |
Publish date | Sep 7, 2015 (structure data deposition date) |
Authors | Milhas, S. / Raux, B. / Betzi, S. / Derviaux, C. / Roche, P. / Restouin, A. / Basse, M.J. / Rebuffet, E. / Lugari, A. / Badol, M. ...Milhas, S. / Raux, B. / Betzi, S. / Derviaux, C. / Roche, P. / Restouin, A. / Basse, M.J. / Rebuffet, E. / Lugari, A. / Badol, M. / Kashyap, R. / Lissitzky, J.C. / Eydoux, C. / Hamon, V. / Gourdel, M.E. / Combes, S. / Zimmermann, P. / Aurrand-Lions, M. / Roux, T. / Rogers, C. / Muller, S. / Knapp, S. / Trinquet, E. / Collette, Y. / Guillemot, J.C. / Morelli, X. |
External links | Acs Chem. Biol. / PubMed:27219844 |
Methods | X-ray diffraction |
Resolution | 1.7 - 1.9 Å |
Structure data | PDB-5dlx: PDB-5dlz: |
Chemicals | ChemComp-5D2: ChemComp-HOH: ChemComp-5D1: |
Source |
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Keywords | TRANSCRIPTION / INHIBITOR / HISTONE / EPIGENETIC READER / BROMODOMAIN / BRD4 / Brd4_BD1 |