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-Structure paper
Title | Discovery of RAF265: A Potent mut-B-RAF Inhibitor for the Treatment of Metastatic Melanoma. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 6, Page 961-965, Year 2015 |
Publish date | Jul 23, 2015 (structure data deposition date) |
Authors | Williams, T.E. / Subramanian, S. / Verhagen, J. / McBride, C.M. / Costales, A. / Sung, L. / Antonios-McCrea, W. / McKenna, M. / Louie, A.K. / Ramurthy, S. ...Williams, T.E. / Subramanian, S. / Verhagen, J. / McBride, C.M. / Costales, A. / Sung, L. / Antonios-McCrea, W. / McKenna, M. / Louie, A.K. / Ramurthy, S. / Levine, B. / Shafer, C.M. / Machajewski, T. / Renhowe, P.A. / Appleton, B.A. / Amiri, P. / Chou, J. / Stuart, D. / Aardalen, K. / Poon, D. |
External links | Acs Med. Chem. Lett. / PubMed:26396681 |
Methods | X-ray diffraction |
Resolution | 3.17 Å |
Structure data | PDB-5ct7: |
Chemicals | ChemComp-55J: |
Source |
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Keywords | TRANSFERASE / kinase |