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-Structure paper
Title | Inhibition of RAF Isoforms and Active Dimers by LY3009120 Leads to Anti-tumor Activities in RAS or BRAF Mutant Cancers. |
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Journal, issue, pages | Cancer Cell, Vol. 28, Page 384-398, Year 2015 |
Publish date | Jun 26, 2015 (structure data deposition date) |
![]() | Peng, S.B. / Henry, J.R. / Kaufman, M.D. / Lu, W.P. / Smith, B.D. / Vogeti, S. / Rutkoski, T.J. / Wise, S. / Chun, L. / Zhang, Y. ...Peng, S.B. / Henry, J.R. / Kaufman, M.D. / Lu, W.P. / Smith, B.D. / Vogeti, S. / Rutkoski, T.J. / Wise, S. / Chun, L. / Zhang, Y. / Van Horn, R.D. / Yin, T. / Zhang, X. / Yadav, V. / Chen, S.H. / Gong, X. / Ma, X. / Webster, Y. / Buchanan, S. / Mochalkin, I. / Huber, L. / Kays, L. / Donoho, G.P. / Walgren, J. / McCann, D. / Patel, P. / Conti, I. / Plowman, G.D. / Starling, J.J. / Flynn, D.L. |
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Methods | X-ray diffraction |
Resolution | 2.7 Å |
Structure data | ![]() PDB-5c9c: |
Chemicals | ![]() ChemComp-4Z5: ![]() ChemComp-CL: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / TRANSFERASE-TRANSFERASE INHIBITOR complex |