+Search query
-Structure paper
Title | Imidazotriazines: Spleen Tyrosine Kinase (Syk) Inhibitors Identified by Free-Energy Perturbation (FEP). |
---|---|
Journal, issue, pages | Chemmedchem, Vol. 11, Page 217-233, Year 2016 |
Publish date | Jun 15, 2015 (structure data deposition date) |
![]() | Lovering, F. / Aevazelis, C. / Chang, J. / Dehnhardt, C. / Fitz, L. / Han, S. / Janz, K. / Lee, J. / Kaila, N. / McDonald, J. ...Lovering, F. / Aevazelis, C. / Chang, J. / Dehnhardt, C. / Fitz, L. / Han, S. / Janz, K. / Lee, J. / Kaila, N. / McDonald, J. / Moore, W. / Moretto, A. / Papaioannou, N. / Richard, D. / Ryan, M.S. / Wan, Z.K. / Thorarensen, A. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.95 - 2.15 Å |
Structure data | ![]() PDB-5c26: ![]() PDB-5c27: |
Chemicals | ![]() ChemComp-50H: ![]() ChemComp-HOH: ![]() ChemComp-50J: ![]() ChemComp-GOL: |
Source |
|
![]() | TRANSFERASE/INHIBITOR / Spleen Tyrosine Kinase / Inhibitor / TRANSFERASE-INHIBITOR complex |