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TitleIdentification of Cyproheptadine as an Inhibitor of SET Domain Containing Lysine Methyltransferase 7/9 (Set7/9) That Regulates Estrogen-Dependent Transcription
Journal, issue, pagesJ. Med. Chem., Vol. 59, Page 3650-3660, Year 2016
Publish dateAug 20, 2015 (structure data deposition date)
AuthorsTakemoto, Y. / Ito, A. / Niwa, H. / Okamura, M. / Fujiwara, T. / Hirano, T. / Handa, N. / Umehara, T. / Sonoda, T. / Ogawa, K. ...Takemoto, Y. / Ito, A. / Niwa, H. / Okamura, M. / Fujiwara, T. / Hirano, T. / Handa, N. / Umehara, T. / Sonoda, T. / Ogawa, K. / Tariq, M. / Nishino, N. / Dan, S. / Kagechika, H. / Yamori, T. / Yokoyama, S. / Yoshida, M.
External linksJ. Med. Chem. / PubMed:27088648
MethodsX-ray diffraction
Resolution2.005 Å
Structure data

PDB-5ayf:
Crystal structure of SET7/9 in complex with cyproheptadine
Method: X-RAY DIFFRACTION / Resolution: 2.005 Å

Chemicals

ChemComp-SAM:
S-ADENOSYLMETHIONINE

ChemComp-C7H:
4-(dibenzo[1,2-a:2',1'-d][7]annulen-11-ylidene)-1-methyl-piperidine / medication*YM

ChemComp-TRS:
2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL / pH buffer*YM

ChemComp-HOH:
WATER

Source
  • homo sapiens (human)
KeywordsTRANSFERASE/TRANSFERASE INHIBITOR / Set domain / methyltransferase / inhibitor / TRANSFERASE-TRANSFERASE INHIBITOR complex

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