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-Structure paper
Title | Crystal Structure of the Bromodomain of Human Surface Epitope Engineered Brd1A in Complex with 3D Consortium Fragment 4-Acetyl-Piperazin-2-One |
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Journal, issue, pages | To be Published |
Publish date | Mar 10, 2015 (structure data deposition date) |
![]() | Pearce, N.M. / Fairhead, M. / Strain-Damerell, C. / Talon, R. / Wright, N. / Ng, J.T. / Bradley, A. / Cox, O. / Bowkett, D. / Collins, P. ...Pearce, N.M. / Fairhead, M. / Strain-Damerell, C. / Talon, R. / Wright, N. / Ng, J.T. / Bradley, A. / Cox, O. / Bowkett, D. / Collins, P. / Brandao-Neto, J. / Douangamath, A. / Krojer, T. / Burgess-Brown, N. / Brennan, P. / Arrowsmith, C.H. / Edwards, E. / Bountra, C. / von Delft, F. |
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Methods | X-ray diffraction |
Resolution | 1.578 Å |
Structure data | ![]() PDB-5ame: |
Chemicals | ![]() ChemComp-PW3: ![]() ChemComp-NA: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSCRIPTION / HISTONE-BINDING PROTEIN / BROMODOMAIN / EPIGENETIC / FRAGMENTSCREENING / STRUCTURAL GENOMICS CONSORTIUM / SGC / DIAMOND I04-1 |