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-Structure paper
Title | Binding mode of the breakthrough inhibitor AZD9291 to epidermal growth factor receptor revealed. |
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Journal, issue, pages | J. Struct. Biol., Vol. 192, Page 539-544, Year 2015 |
Publish date | Apr 14, 2015 (structure data deposition date) |
![]() | Yosaatmadja, Y. / Silva, S. / Dickson, J.M. / Patterson, A.V. / Smaill, J.B. / Flanagan, J.U. / McKeage, M.J. / Squire, C.J. |
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Methods | X-ray diffraction |
Resolution | 2.8 Å |
Structure data | ![]() PDB-4zau: |
Chemicals | ![]() ChemComp-YY3: ![]() ChemComp-HOH: |
Source |
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![]() | transferase/transferase inhibitor / transferase / kinase domain / transferase-transferase inhibitor complex |