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-Structure paper
Title | Regulatory T Cell Modulation by CBP/EP300 Bromodomain Inhibition. |
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Journal, issue, pages | J. Biol. Chem., Vol. 291, Page 13014-13027, Year 2016 |
Publish date | Mar 3, 2015 (structure data deposition date) |
![]() | Ghosh, S. / Taylor, A. / Chin, M. / Huang, H.R. / Conery, A.R. / Mertz, J.A. / Salmeron, A. / Dakle, P.J. / Mele, D. / Cote, A. ...Ghosh, S. / Taylor, A. / Chin, M. / Huang, H.R. / Conery, A.R. / Mertz, J.A. / Salmeron, A. / Dakle, P.J. / Mele, D. / Cote, A. / Jayaram, H. / Setser, J.W. / Poy, F. / Hatzivassiliou, G. / DeAlmeida-Nagata, D. / Sandy, P. / Hatton, C. / Romero, F.A. / Chiang, E. / Reimer, T. / Crawford, T. / Pardo, E. / Watson, V.G. / Tsui, V. / Cochran, A.G. / Zawadzke, L. / Harmange, J.C. / Audia, J.E. / Bryant, B.M. / Cummings, R.T. / Magnuson, S.R. / Grogan, J.L. / Bellon, S.F. / Albrecht, B.K. / Sims, R.J. / Lora, J.M. |
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Methods | X-ray diffraction |
Resolution | 1.65 - 1.86 Å |
Structure data | ![]() PDB-4yk0: ![]() PDB-5dbm: |
Chemicals | ![]() ChemComp-986: ![]() ChemComp-EDO: ![]() ChemComp-HOH: ![]() ChemComp-58N: |
Source |
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![]() | TRANSFERASE / CBP / CPI098 / PROTEIN BINDING / bromodomain / inhibitor / epigenetics / chromatin |