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-Structure paper
Title | RAF inhibitors that evade paradoxical MAPK pathway activation. |
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Journal, issue, pages | Nature, Vol. 526, Page 583-586, Year 2015 |
Publish date | Jan 26, 2015 (structure data deposition date) |
![]() | Zhang, C. / Spevak, W. / Zhang, Y. / Burton, E.A. / Ma, Y. / Habets, G. / Zhang, J. / Lin, J. / Ewing, T. / Matusow, B. ...Zhang, C. / Spevak, W. / Zhang, Y. / Burton, E.A. / Ma, Y. / Habets, G. / Zhang, J. / Lin, J. / Ewing, T. / Matusow, B. / Tsang, G. / Marimuthu, A. / Cho, H. / Wu, G. / Wang, W. / Fong, D. / Nguyen, H. / Shi, S. / Womack, P. / Nespi, M. / Shellooe, R. / Carias, H. / Powell, B. / Light, E. / Sanftner, L. / Walters, J. / Tsai, J. / West, B.L. / Visor, G. / Rezaei, H. / Lin, P.S. / Nolop, K. / Ibrahim, P.N. / Hirth, P. / Bollag, G. |
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Methods | X-ray diffraction |
Resolution | 2 - 2.8 Å |
Structure data | ![]() PDB-4xv1: ![]() PDB-4xv2: ![]() PDB-4xv3: ![]() PDB-4xv9: |
Chemicals | ![]() ChemComp-904: ![]() ChemComp-HOH: ![]() ChemComp-P06: ![]() ChemComp-P02: ![]() ChemComp-1OO: ![]() ChemComp-SO4: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / ![]() ![]() ![]() ![]() ![]() |