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-Structure paper
Title | Discovery of highly potent, selective, and efficacious small molecule inhibitors of ERK1/2. |
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Journal, issue, pages | J. Med. Chem., Vol. 58, Page 1976-1991, Year 2015 |
Publish date | Jan 8, 2015 (structure data deposition date) |
![]() | Ren, L. / Grina, J. / Moreno, D. / Blake, J.F. / Gaudino, J.J. / Garrey, R. / Metcalf, A.T. / Burkard, M. / Martinson, M. / Rasor, K. ...Ren, L. / Grina, J. / Moreno, D. / Blake, J.F. / Gaudino, J.J. / Garrey, R. / Metcalf, A.T. / Burkard, M. / Martinson, M. / Rasor, K. / Chen, H. / Dean, B. / Gould, S.E. / Pacheco, P. / Shahidi-Latham, S. / Yin, J. / West, K. / Wang, W. / Moffat, J.G. / Schwarz, J.B. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.58 Å |
Structure data | ![]() PDB-4xj0: |
Chemicals | ![]() ChemComp-41B: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / protein Kinase / TRANSFERASE-TRANSFERASE INHIBITOR complex |