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-Structure paper
Title | LLY-507, a Cell-active, Potent, and Selective Inhibitor of Protein-lysine Methyltransferase SMYD2. |
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Journal, issue, pages | J. Biol. Chem., Vol. 290, Page 13641-13653, Year 2015 |
Publish date | Nov 4, 2014 (structure data deposition date) |
![]() | Nguyen, H. / Allali-Hassani, A. / Antonysamy, S. / Chang, S. / Chen, L.H. / Curtis, C. / Emtage, S. / Fan, L. / Gheyi, T. / Li, F. ...Nguyen, H. / Allali-Hassani, A. / Antonysamy, S. / Chang, S. / Chen, L.H. / Curtis, C. / Emtage, S. / Fan, L. / Gheyi, T. / Li, F. / Liu, S. / Martin, J.R. / Mendel, D. / Olsen, J.B. / Pelletier, L. / Shatseva, T. / Wu, S. / Zhang, F.F. / Arrowsmith, C.H. / Brown, P.J. / Campbell, R.M. / Garcia, B.A. / Barsyte-Lovejoy, D. / Mader, M. / Vedadi, M. |
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Methods | X-ray diffraction |
Resolution | 1.63 Å |
Structure data | ![]() PDB-4wuy: |
Chemicals | ![]() ChemComp-3UJ: ![]() ChemComp-SAH: ![]() ChemComp-GOL: ![]() ChemComp-ZN: ![]() ChemComp-HOH: |
Source |
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![]() | Transferase/transferase inhibitor / SMYD2 - LLY-507 / Transferase-transferase inhibitor complex |