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-Structure paper
Title | A reversed sulfonamide series of selective RORc inverse agonists. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 24, Page 5769-5776, Year 2014 |
Publish date | Oct 7, 2014 (structure data deposition date) |
Authors | van Niel, M.B. / Fauber, B.P. / Cartwright, M. / Gaines, S. / Killen, J.C. / Rene, O. / Ward, S.I. / de Leon Boenig, G. / Deng, Y. / Eidenschenk, C. ...van Niel, M.B. / Fauber, B.P. / Cartwright, M. / Gaines, S. / Killen, J.C. / Rene, O. / Ward, S.I. / de Leon Boenig, G. / Deng, Y. / Eidenschenk, C. / Everett, C. / Gancia, E. / Ganguli, A. / Gobbi, A. / Hawkins, J. / Johnson, A.R. / Kiefer, J.R. / La, H. / Lockey, P. / Norman, M. / Ouyang, W. / Qin, A. / Wakes, N. / Waszkowycz, B. / Wong, H. |
External links | Bioorg. Med. Chem. Lett. / PubMed:25453817 |
Methods | X-ray diffraction |
Resolution | 1.702 Å |
Structure data | PDB-4wlb: |
Chemicals | ChemComp-3QQ: ChemComp-TLA: ChemComp-HOH: |
Source |
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Keywords | TRANSCRIPTION / NUCLEAR RECEPTOR LIGAND BINDING DOMAIN |